Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50018328
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50035696(AMD-3100 | CHEMBL18442 | 11-{4-[4,8, 11-1,4,8,11te...)
Affinity DataIC50: 2.90nMAssay Description:Antagonist activity at CXCR4 receptor in SDF-1alpha-stimulated human SUP-T1 cells incubated for 30 mins by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421849(CHEMBL5283078)
Affinity DataIC50: 20nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421854(CHEMBL5269411)
Affinity DataIC50: 41nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421857(CHEMBL5290852)
Affinity DataIC50: 48nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421853(CHEMBL5282178)
Affinity DataIC50: 68nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421860(CHEMBL5283630)
Affinity DataIC50: 68nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421856(CHEMBL5277914)
Affinity DataIC50: 69nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421859(CHEMBL5285076)
Affinity DataIC50: 81nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421849(CHEMBL5283078)
Affinity DataIC50: 119nMAssay Description:Antagonist activity at CXCR4 receptor in SDF-1alpha-stimulated human SUP-T1 cells incubated for 30 mins by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421861(CHEMBL5275975)
Affinity DataIC50: 119nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421863(CHEMBL5277386)
Affinity DataIC50: 122nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421858(CHEMBL5276826)
Affinity DataIC50: 147nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421852(CHEMBL5283007)
Affinity DataIC50: 156nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421862(CHEMBL5291454)
Affinity DataIC50: 194nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421851(CHEMBL5273456)
Affinity DataIC50: 312nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50035696(AMD-3100 | CHEMBL18442 | 11-{4-[4,8, 11-1,4,8,11te...)
Affinity DataIC50: 325nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421855(CHEMBL5266216)
Affinity DataIC50: 354nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetStromal cell-derived factor 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50035696(AMD-3100 | CHEMBL18442 | 11-{4-[4,8, 11-1,4,8,11te...)
Affinity DataIC50: 608nMAssay Description:Inhibition of SDF-1 alpha induced cell migration in human SUP-T1 cells pre-incubated for 30 mins followed by SDF-1 alpha addition measured after 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetStromal cell-derived factor 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421849(CHEMBL5283078)
Affinity DataIC50: 621nMAssay Description:Inhibition of SDF-1 alpha induced cell migration in human SUP-T1 cells pre-incubated for 30 mins followed by SDF-1 alpha addition measured after 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421848(CHEMBL5278283)
Affinity DataIC50: 699nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421864(CHEMBL5283015)
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM194537(US9205085, MSX- 161s)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 4(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50421850(CHEMBL5280629)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to CXCR4 (unknown origin) expressed in CHO cells incubated for 40 mins by competitive binding assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed