Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50010659
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540865(CHEMBL4640012)
Affinity DataIC50: 0.430nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540872(CHEMBL4647222)
Affinity DataIC50: 1nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50187686(CHEMBL3828074 | US9670204, 2 2-((2-ethyl-6-(4-(2-(...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50187693(CHEMBL3186509)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50187693(CHEMBL3186509)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human ATX by fluorogenic substrate-3 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540884(CHEMBL4644036)
Affinity DataIC50: 16nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540863(CHEMBL4641011)
Affinity DataIC50: 21nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540862(CHEMBL4639039)
Affinity DataIC50: 31nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540873(CHEMBL4643433)
Affinity DataIC50: 34nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540867(CHEMBL4633587)
Affinity DataIC50: 35nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540870(CHEMBL4643937)
Affinity DataIC50: 37nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50264199(CHEMBL4086925)
Affinity DataIC50: 60nMAssay Description:Inhibition of human ATX by LPC choline release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540864(CHEMBL4644515)
Affinity DataIC50: 63nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540887(CHEMBL4634620)
Affinity DataIC50: 69nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540886(CHEMBL4638125)
Affinity DataIC50: 107nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540877(CHEMBL4644727)
Affinity DataIC50: 117nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540871(CHEMBL4636755)
Affinity DataIC50: 122nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540874(CHEMBL4638854)
Affinity DataIC50: 127nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540868(CHEMBL4637219)
Affinity DataIC50: 127nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50187686(CHEMBL3828074 | US9670204, 2 2-((2-ethyl-6-(4-(2-(...)
Affinity DataIC50: 131nMAssay Description:Inhibition of human ATX by LPC choline release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540882(CHEMBL4636225)
Affinity DataIC50: 135nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540888(CHEMBL4639826)
Affinity DataIC50: 180nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540869(CHEMBL4634766)
Affinity DataIC50: 199nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540875(CHEMBL4643457)
Affinity DataIC50: 210nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540881(CHEMBL4643989)
Affinity DataIC50: 231nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540866(CHEMBL4642973)
Affinity DataIC50: 297nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM555294(BDBM50540913 | 34(6-chloro-2-cyclopropyl-1-(1-(eth...)
Affinity DataIC50: 500nMAssay Description:Inhibition of human ATX by LPC choline release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540880(CHEMBL4646372)
Affinity DataIC50: 508nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540883(CHEMBL4637140)
Affinity DataIC50: 610nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540878(CHEMBL4635930)
Affinity DataIC50: 613nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540885(CHEMBL4640212)
Affinity DataIC50: 655nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540912(CHEMBL4636797)
Affinity DataIC50: 740nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540901(CHEMBL4645651)
Affinity DataIC50: 757nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540890(CHEMBL4647615)
Affinity DataIC50: 879nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540889(CHEMBL4643078)
Affinity DataIC50: 906nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540876(CHEMBL4641104)
Affinity DataIC50: 970nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540904(CHEMBL4644717)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540879(CHEMBL4636002)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540898(CHEMBL4635487)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540911(CHEMBL4648648)
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540905(CHEMBL4649805)
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540906(CHEMBL4641845)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540896(CHEMBL4636052)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540908(CHEMBL4635805)
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540897(CHEMBL4644862)
Affinity DataIC50: 2.31E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540902(CHEMBL4637835)
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540903(CHEMBL4645284)
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540895(CHEMBL4634132)
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540907(CHEMBL4634398)
Affinity DataIC50: 3.96E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAutotaxin(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540892(CHEMBL4642425)
Affinity DataIC50: 5.24E+3nMAssay Description:Inhibition of human ATX pre-incubated for 45 mins before fluorogenic substrate-3 addition and measured every minute for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
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