Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50010857
TargetSolute carrier organic anion transporter family member 1B3(Human)
University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50542676(CHEMBL4633668)
Affinity DataEC50:  3nMAssay Description:Substrate activity at OATP1B3 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B3(Human)
University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50542677(CHEMBL4637446)
Affinity DataEC50:  2.40nMAssay Description:Substrate activity at OATP1B3 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B3(Human)
University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50542678(CHEMBL4636474)
Affinity DataEC50:  1.40nMAssay Description:Substrate activity at OATP1B3 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50542676(CHEMBL4633668)
Affinity DataEC50:  4.5nMAssay Description:Substrate activity at OATP1B1 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50542677(CHEMBL4637446)
Affinity DataEC50:  1.10nMAssay Description:Substrate activity at OATP1B1 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
University of Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50542678(CHEMBL4636474)
Affinity DataEC50:  1.70nMAssay Description:Substrate activity at OATP1B1 (unknown origin) expressed in HEK293 cells assessed as cytotoxicity incubated for 48 hrs by sulforhodamine B assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed