Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50010650
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50003020(MK-3102 | OMARIGLIPTIN | US10155775, Omarigliptin ...)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540854(CHEMBL4641763)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540853(CHEMBL4644314)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540856(CHEMBL4636223)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540851(CHEMBL4640183)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540852(CHEMBL4634272)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540858(CHEMBL4640418)
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540855(CHEMBL4634474)
Affinity DataIC50: 27nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540850(CHEMBL4635433)
Affinity DataIC50: 49nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540857(CHEMBL4649110)
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540847(CHEMBL4635648)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540848(CHEMBL4633377)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540849(CHEMBL4643841)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG by manual whole-cell patch-clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A5(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 4.58E+4nMAssay Description:Inhibition of recombinant human CYP3A5 using midazolam as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 4.58E+4nMAssay Description:Inhibition of recombinant human CYP3A4 using midazolam as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 7.63E+4nMAssay Description:Inhibition of recombinant human CYP2C8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2E1(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2E1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant DPP9 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant DPP8 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A4 using testosterone as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A5(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A5 using testosterone as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A4 using midazolam as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A5(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A5 using midazolam as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2A6(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2A6More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2B6(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2B6More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C19More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2E1(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2E1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A4 using testosterone as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A5(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A5 using testosterone as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A5(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A5 using testosterone as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C19More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2B6(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2B6More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2A6(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2A6More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP1A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A5(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A5 using midazolam as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A4 using midazolam as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A4 using testosterone as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2E1(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2E1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C19More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
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