Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50010423
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50075103(CHEBI:48202 | Nanafrocin)
Affinity DataIC50: 500nMAssay Description:Inhibition of human DNMT3B using [3H]-SAMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50075103(CHEBI:48202 | Nanafrocin)
Affinity DataIC50: 730nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells by DRONE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50389497(CHEMBL1564869)
Affinity DataIC50: 900nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50075103(CHEBI:48202 | Nanafrocin)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538703(CHEMBL4645141)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells by DRONE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538703(CHEMBL4645141)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538702(CHEMBL4634562)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538701(CHEMBL4647360)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538691(CHEMBL4640870)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538695(CHEMBL4642475)
Affinity DataIC50: 2.24E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 1(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538691(CHEMBL4640870)
Affinity DataIC50: 2.72E+4nMAssay Description:Inhibition of human recombinant DNMT1 expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucle...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538700(CHEMBL4647309)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 1(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538692(CHEMBL4649221)
Affinity DataIC50: 2.85E+4nMAssay Description:Inhibition of human recombinant DNMT1 expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucle...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538696(CHEMBL4642377)
Affinity DataIC50: 3.72E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538699(CHEMBL4637965)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538694(CHEMBL4647111)
Affinity DataIC50: 6.68E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538697(CHEMBL4641323)
Affinity DataIC50: 7.04E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538693(CHEMBL4632355)
Affinity DataIC50: 7.23E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3B(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50538698(CHEMBL4644275)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human recombinant DNMT3B expressed in baculovirus infected insect cells using CpG site containing internally quenched hairpin oligonucl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed