Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50010621
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540648BDBM50540648(CHEMBL4639944)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540643BDBM50540643(CHEMBL4639941)
Affinity DataIC50: 0.130nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540639BDBM50540639(CHEMBL4632810)
Affinity DataIC50: 0.130nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540640BDBM50540640(CHEMBL4641768)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540649BDBM50540649(CHEMBL4642214)
Affinity DataIC50: 0.160nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540655BDBM50540655(CHEMBL4635889)
Affinity DataIC50: 0.170nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540642BDBM50540642(CHEMBL4649085)
Affinity DataIC50: 0.180nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540644BDBM50540644(CHEMBL4639413)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540638BDBM50540638(CHEMBL4649563)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540645BDBM50540645(CHEMBL4645937)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540646BDBM50540646(CHEMBL4634153)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540654BDBM50540654(CHEMBL4642738)
Affinity DataIC50: 0.270nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540653BDBM50540653(CHEMBL4637660)
Affinity DataIC50: 0.280nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540641BDBM50540641(CHEMBL4636234)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540651BDBM50540651(CHEMBL4645131)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540652BDBM50540652(CHEMBL4638582)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540647BDBM50540647(CHEMBL4641915)
Affinity DataIC50: 0.380nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540650BDBM50540650(CHEMBL4640188)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540656BDBM50540656(CHEMBL4644376)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540659BDBM50540659(CHEMBL4646883)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540637BDBM50540637(CHEMBL4647151)
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540657BDBM50540657(CHEMBL4642447)
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540658BDBM50540658(CHEMBL4648160)
Affinity DataIC50: 2.29E+3nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540660BDBM50540660(CHEMBL4644683)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540636BDBM50540636(CHEMBL4647625)
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236398BDBM50236398(CHEMBL1503273)
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540662BDBM50540662(CHEMBL4639754)
Affinity DataIC50: 3.04E+4nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540667BDBM50540667(CHEMBL4639402)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540666BDBM50540666(CHEMBL4641231)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540665BDBM50540665(CHEMBL4647974)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540664BDBM50540664(CHEMBL4643702)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540663BDBM50540663(CHEMBL4646647)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540661BDBM50540661(CHEMBL4639446)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed