Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50010605
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540553BDBM50540553(CHEMBL4644726)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540555BDBM50540555(CHEMBL4642691)
Affinity DataIC50: 210nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540566BDBM50540566(CHEMBL4636567)
Affinity DataIC50: 240nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540554BDBM50540554(CHEMBL4636810)
Affinity DataIC50: 330nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540556BDBM50540556(CHEMBL4636520)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540552BDBM50540552(CHEMBL4636990)
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540557BDBM50540557(CHEMBL4642679)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540571BDBM50540571(CHEMBL4632967)
Affinity DataIC50: 1.52E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540568BDBM50540568(CHEMBL4634884)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540561BDBM50540561(CHEMBL4643748)
Affinity DataIC50: 2.67E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540562BDBM50540562(CHEMBL4649566)
Affinity DataIC50: 2.72E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540558BDBM50540558(CHEMBL4641671)
Affinity DataIC50: 2.80E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540560BDBM50540560(CHEMBL4635054)
Affinity DataIC50: 2.98E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540559BDBM50540559(CHEMBL4638499)
Affinity DataIC50: 3.20E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540567BDBM50540567(CHEMBL4647531)
Affinity DataIC50: 3.32E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540569BDBM50540569(CHEMBL4635727)
Affinity DataIC50: 6.10E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540563BDBM50540563(CHEMBL4644539)
Affinity DataIC50: 7.00E+3nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540570BDBM50540570(CHEMBL4639127)
Affinity DataIC50: 1.03E+4nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540565BDBM50540565(CHEMBL4641643)
Affinity DataIC50: 1.21E+4nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540564BDBM50540564(CHEMBL4648827)
Affinity DataIC50: 1.23E+4nMAssay Description:Antagonist activity at GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
"G. D'Annunzio" University of Chieti-Pescara

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540552BDBM50540552(CHEMBL4636990)
Affinity DataIC50: 1.40E+4nMAssay Description:Antagonist activity at GAL4-tagged human PPARgamma LBD expressed in human HepG2 cells assessed as inhibition of Wy14,643-induced receptor transactiva...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed