Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50010962
TargetAurora kinase A(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50004231(CHEMBL3237167)
Affinity DataIC50: 5nMAssay Description:Inhibition of AURKA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543797(CHEMBL4637300)
Affinity DataIC50: 90nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM14210(N-[4-({6-methoxy-7-[3-(morpholin-4-yl)propoxy]quin...)
Affinity DataIC50: 110nMAssay Description:Inhibition of AURKA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM14210(N-[4-({6-methoxy-7-[3-(morpholin-4-yl)propoxy]quin...)
Affinity DataIC50: 130nMAssay Description:Inhibition of AURKB (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543797(CHEMBL4637300)
Affinity DataIC50: 930nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543800(CHEMBL4645713)
Affinity DataIC50: 980nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543799(CHEMBL4640153)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543801(CHEMBL4648901)
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543799(CHEMBL4640153)
Affinity DataIC50: 1.77E+3nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543800(CHEMBL4645713)
Affinity DataIC50: 2.99E+3nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543796(CHEMBL4635411)
Affinity DataIC50: 6.89E+3nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543796(CHEMBL4635411)
Affinity DataIC50: 7.64E+3nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543802(CHEMBL4644959)
Affinity DataIC50: 8.33E+3nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543803(CHEMBL4639147)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543795(CHEMBL4645551)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543798(CHEMBL4641064)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of human Aurora B using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543798(CHEMBL4641064)
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50543795(CHEMBL4645551)
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of human Aurora A using [H-LRRASLG] as substrate in presence of [gamma-33P]-ATP incubated for 2 hrs by hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed