Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50010954
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50457446(CHEMBL4212692)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM221688(US9314464, 9 | US9593100, Compound 9 | US10568884,...)
Affinity DataIC50: 4nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM25617(N-[3-({5-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl}carb...)
Affinity DataIC50: 13nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 22nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50396483(PLX-4032 | RG 7204 | Ro 5185426 | VEMURAFENIB | US...)
Affinity DataIC50: 31nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50096279(CHEMBL3577124)
Affinity DataIC50: 31nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50543733(CHEMBL4644256)
Affinity DataIC50: 80nMAssay Description:Inhibition of human BRAF V600E mutant by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50543732(CHEMBL4640613)
Affinity DataIC50: 85nMAssay Description:Inhibition of human BRAF V600E mutant by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50543731(CHEMBL4644507)
Affinity DataIC50: 114nMAssay Description:Inhibition of human BRAF V600E mutant by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50543726(CHEMBL4649497)
Affinity DataIC50: 350nMAssay Description:Inhibition of human BRAF V600E mutant by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50543730(CHEMBL4646680)
Affinity DataIC50: 500nMAssay Description:Inhibition of human BRAF V600E mutant by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50543724(CHEMBL4638623)
Affinity DataIC50: 750nMAssay Description:Inhibition of human BRAF V600E mutant by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50543727(CHEMBL4641369)
Affinity DataIC50: 790nMAssay Description:Inhibition of human BRAF V600E mutant by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50543725(CHEMBL4646182)
Affinity DataIC50: 880nMAssay Description:Inhibition of human BRAF V600E mutant by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50543729(CHEMBL4641994)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human BRAF V600E mutant by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
National Research Centre (Nrc Id: 60014618)

Curated by ChEMBL
LigandPNGBDBM50543728(CHEMBL4645995)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human BRAF V600E mutant by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed