Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50010951
TargetCysteine proteinase B(Leishmania mexicana)
Universidade De Mogi Das Cruzes (Umc)

Curated by ChEMBL
LigandPNGBDBM50543686(CHEMBL4640351)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of Leishmania mexicana rCPB2.8 using Z-FR-AMC as substrate by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Universidade De Mogi Das Cruzes (Umc)

Curated by ChEMBL
LigandPNGBDBM50543685(CHEMBL4640915)
Affinity DataIC50: 3.69E+3nMAssay Description:Inhibition of cathepsin L (unknown origin) using Z-FR-AMC as substrate by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCathepsin B(Human)
Universidade De Mogi Das Cruzes (Umc)

Curated by ChEMBL
LigandPNGBDBM50543685(CHEMBL4640915)
Affinity DataIC50: 6.86E+3nMAssay Description:Inhibition of cathepsin B (unknown origin) using Z-FR-AMC as substrate by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCysteine proteinase B(Leishmania mexicana)
Universidade De Mogi Das Cruzes (Umc)

Curated by ChEMBL
LigandPNGBDBM50543687(CHEMBL4636701)
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of Leishmania mexicana rCPB2.8 using Z-FR-AMC as substrate by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCysteine proteinase B(Leishmania mexicana)
Universidade De Mogi Das Cruzes (Umc)

Curated by ChEMBL
LigandPNGBDBM50543688(CHEMBL4635812)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of Leishmania mexicana rCPB2.8 using Z-FR-AMC as substrate by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCysteine proteinase B(Leishmania mexicana)
Universidade De Mogi Das Cruzes (Umc)

Curated by ChEMBL
LigandPNGBDBM50543686(CHEMBL4640351)
Affinity DataKi:  2.17E+4nMAssay Description:Inhibition of Leishmania mexicana rCPB2.8 assessed as inhibition constant using Z-FR-AMC as substrate preincubated for 10 mins followed by substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed