Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50011187
TargetHistone deacetylase 6(Human)
Cedilla Therapeutics

Curated by ChEMBL
LigandPNGBDBM50507688(CHEMBL4550214 | US11535598, Compound 5)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProtein phosphatase 1 regulatory subunit 15B(Human)
Cedilla Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545524(CHEMBL2369159)
Affinity DataIC50: 33nMAssay Description:Inhibition of amino-terminal MBP-tagged/carboxy-terminal His6-tagged human PPP1R15B (325 to 626 residues)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Cedilla Therapeutics

Curated by ChEMBL
LigandPNGBDBM50507688(CHEMBL4550214 | US11535598, Compound 5)
Affinity DataIC50: 200nMAssay Description:Inhibition of MELK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Cedilla Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545524(CHEMBL2369159)
Affinity DataIC50: 200nMAssay Description:Inhibition of MELK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Cedilla Therapeutics

Curated by ChEMBL
LigandPNGBDBM50043341(CHEMBL3355059)
Affinity DataIC50: 200nMAssay Description:Inhibition of MELK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Cedilla Therapeutics

Curated by ChEMBL
LigandPNGBDBM50466857(CHEMBL4288096)
Affinity DataIC50: 200nMAssay Description:Inhibition of MELK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Cedilla Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545525(CHEMBL4640049)
Affinity DataIC50: 200nMAssay Description:Inhibition of MELK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProtein phosphatase 1 regulatory subunit 15A(Human)
Cedilla Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545524(CHEMBL2369159)
Affinity DataIC50: 977nMAssay Description:Inhibition of amino-terminal MBP-tagged/carboxy-terminal His6-tagged human PPP1R15A (325 to 626 residues)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed