Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50012725
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Inhibition of VGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human HDAC1 expressed in baculovirus expression system using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate after 24 hrs ...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human HDAC3 expressed in baculovirus expression system using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate after 24 hrs ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 225nMAssay Description:Inhibition of BRD4 BD2 domain (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 291nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of recombinant human HDAC6 expressed in baculovirus expression system using Ac-Lys-Tyr-Lys (epsilon-acetyl)-AMC as substrate after 24 hrs ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Shandong First Medical University & Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair



































3D Structure (crystal)



