Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50010846
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Central South University
Curated by ChEMBL
Central South University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human PI3K p110delta by HTRF assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Central South University
Curated by ChEMBL
Central South University
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of human PI3K (p110alpha/p85alpha) by HTRF assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Central South University
Curated by ChEMBL
Central South University
Curated by ChEMBL
Affinity DataIC50: 119nMAssay Description:Inhibition of human PI3K p110delta by HTRF assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Central South University
Curated by ChEMBL
Central South University
Curated by ChEMBL
Affinity DataIC50: 122nMAssay Description:Inhibition of human PI3K (p110alpha/p85alpha) by HTRF assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Central South University
Curated by ChEMBL
Central South University
Curated by ChEMBL
Affinity DataIC50: 324nMAssay Description:Inhibition of human PI3K p110beta by HTRF assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Central South University
Curated by ChEMBL
Central South University
Curated by ChEMBL
Affinity DataIC50: 663nMAssay Description:Inhibition of human PI3K p110gamma by HTRF assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Central South University
Curated by ChEMBL
Central South University
Curated by ChEMBL
Affinity DataIC50: 746nMAssay Description:Inhibition of human PI3K p110gamma by HTRF assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Central South University
Curated by ChEMBL
Central South University
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human PI3K p110beta by HTRF assayMore data for this Ligand-Target Pair

