Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50010844
TargetSerine/threonine-protein kinase haspin(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50542441(CHEMBL4642838)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant Haspin (470 to 798 residues) expressed in bacteria using Histone H3 and ARTKQTARKSTGGKAPRKQLA as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50542439(CHEMBL4637707)
Affinity DataIC50: 77nMAssay Description:Inhibition of human recombinant Haspin (470 to 798 residues) expressed in bacteria using Histone H3 and ARTKQTARKSTGGKAPRKQLA as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50542438(CHEMBL4647459)
Affinity DataIC50: 424nMAssay Description:Inhibition of human recombinant CDK9/Cyclin T expressed in baculovirus in Sf9 insect cells using SPTSPSYSPTSPSYSPTSPSKKKK as substrate in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50542439(CHEMBL4637707)
Affinity DataIC50: 495nMAssay Description:Inhibition of human recombinant CDK9/Cyclin T expressed in baculovirus in Sf9 insect cells using SPTSPSYSPTSPSYSPTSPSKKKK as substrate in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50542438(CHEMBL4647459)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of human recombinant Haspin (470 to 798 residues) expressed in bacteria using Histone H3 and ARTKQTARKSTGGKAPRKQLA as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
North-West University

Curated by ChEMBL
LigandPNGBDBM50542440(CHEMBL4634490)
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of human recombinant Haspin (470 to 798 residues) expressed in bacteria using Histone H3 and ARTKQTARKSTGGKAPRKQLA as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed