Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50009353
TargetCREB-binding protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527820(CHEMBL4549898)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to recombinant CBP (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527823(CHEMBL4517875)
Affinity DataKd:  2.63E+3nMAssay Description:Binding affinity to recombinant BRD3 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527820(CHEMBL4549898)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to recombinant BRD2 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)
Affinity DataKd:  886nMAssay Description:Binding affinity to recombinant BRD2 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)
Affinity DataKd:  718nMAssay Description:Binding affinity to recombinant BRD4 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  92nMAssay Description:Binding affinity to recombinant BRD4 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  1.14E+3nMAssay Description:Binding affinity to recombinant BRD4 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  9.60E+3nMAssay Description:Binding affinity to recombinant CBP (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527821(CHEMBL4455209)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to recombinant CBP (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  81nMAssay Description:Binding affinity to recombinant BRD3 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)
Affinity DataKd:  3.18E+3nMAssay Description:Binding affinity to recombinant BRDT BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527823(CHEMBL4517875)
Affinity DataKd:  2.55E+3nMAssay Description:Binding affinity to recombinant BRDT BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  708nMAssay Description:Binding affinity to recombinant BRDT BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  183nMAssay Description:Binding affinity to recombinant BRDT BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)
Affinity DataKd:  84nMAssay Description:Binding affinity to recombinant BRD4 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527820(CHEMBL4549898)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to recombinant BRDT BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to recombinant BRD3 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527823(CHEMBL4517875)
Affinity DataKd:  2.77E+3nMAssay Description:Binding affinity to recombinant BRDT BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  4.84E+3nMAssay Description:Binding affinity to recombinant BRDT BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)
Affinity DataKd:  3.59E+3nMAssay Description:Binding affinity to recombinant BRDT BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527821(CHEMBL4455209)
Affinity DataKd:  2.32E+3nMAssay Description:Binding affinity to recombinant BRDT BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527823(CHEMBL4517875)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to recombinant CBP (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527823(CHEMBL4517875)
Affinity DataKd:  127nMAssay Description:Binding affinity to recombinant BRD4 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  135nMAssay Description:Binding affinity to recombinant BRD4 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 2(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527821(CHEMBL4455209)
Affinity DataKd:  791nMAssay Description:Binding affinity to recombinant BRD2 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527820(CHEMBL4549898)
Affinity DataKd:  1.72E+3nMAssay Description:Binding affinity to recombinant BRD3 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527821(CHEMBL4455209)
Affinity DataKd:  2.87E+3nMAssay Description:Binding affinity to recombinant BRDT BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to recombinant CBP (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527823(CHEMBL4517875)
Affinity DataKd:  139nMAssay Description:Binding affinity to recombinant BRD4 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527821(CHEMBL4455209)
Affinity DataKd:  845nMAssay Description:Binding affinity to recombinant BRD2 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  69nMAssay Description:Binding affinity to recombinant BRD3 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  217nMAssay Description:Binding affinity to recombinant BRDT BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  52nMAssay Description:Binding affinity to recombinant BRD2 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  203nMAssay Description:Binding affinity to recombinant BRD3 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527820(CHEMBL4549898)
Affinity DataKd:  1.21E+3nMAssay Description:Binding affinity to recombinant BRD2 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to recombinant CBP (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  3.96E+3nMAssay Description:Binding affinity to recombinant BRD3 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527821(CHEMBL4455209)
Affinity DataKd:  2.08E+3nMAssay Description:Binding affinity to recombinant BRD3 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527820(CHEMBL4549898)
Affinity DataKd:  2.41E+3nMAssay Description:Binding affinity to recombinant BRDT BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527820(CHEMBL4549898)
Affinity DataKd:  86nMAssay Description:Binding affinity to recombinant BRD4 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527821(CHEMBL4455209)
Affinity DataKd:  67nMAssay Description:Binding affinity to recombinant BRD4 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527820(CHEMBL4549898)
Affinity DataKd:  93nMAssay Description:Binding affinity to recombinant BRD4 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527821(CHEMBL4455209)
Affinity DataKd:  684nMAssay Description:Binding affinity to recombinant BRD4 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  62nMAssay Description:Binding affinity to recombinant BRD4 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527823(CHEMBL4517875)
Affinity DataKd:  1.96E+3nMAssay Description:Binding affinity to recombinant BRD3 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)
Affinity DataKd:  3.12E+3nMAssay Description:Binding affinity to recombinant BRD3 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  5.78E+3nMAssay Description:Binding affinity to recombinant BRD2 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 2(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50527823(CHEMBL4517875)
Affinity DataKd:  1.29E+3nMAssay Description:Binding affinity to recombinant BRD2 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  78nMAssay Description:Binding affinity to recombinant BRD2 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataKd:  251nMAssay Description:Binding affinity to recombinant BRD2 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
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