Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50008003
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50514785(CHEMBL4443903)
Affinity DataKd:  2.40nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50514786(CHEMBL4541406)
Affinity DataKd:  14nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50514787(CHEMBL4449322)
Affinity DataKd:  7.30nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50514788(CHEMBL4440761)
Affinity DataKd:  2.70nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50457446(CHEMBL4212692)
Affinity DataKd:  0.330nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50396483(PLX-4032 | RG 7204 | Ro 5185426 | VEMURAFENIB | US...)
Affinity DataKd:  51nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50514788(CHEMBL4440761)
Affinity DataKd:  2.60nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50457446(CHEMBL4212692)
Affinity DataKd:  0.370nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50514786(CHEMBL4541406)
Affinity DataKd:  9.5nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50514785(CHEMBL4443903)
Affinity DataKd:  2nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50514787(CHEMBL4449322)
Affinity DataKd:  5.10nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cullgen

Curated by ChEMBL
LigandPNGBDBM50396483(PLX-4032 | RG 7204 | Ro 5185426 | VEMURAFENIB | US...)
Affinity DataKd:  58nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed