Compile Data Set for Download or QSAR
Report error Found 203 Enz. Inhib. hit(s) with all data for entry = 50018471
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470579BDBM50470579(4sc-202 | Domatinostat)
Affinity DataIC50: 0.160nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470576BDBM50470576(CHEMBL4294949)
Affinity DataIC50: 0.160nMAssay Description:Inhibition of human recombinant HDAC3 at 0.5 uM using Fluor-de-Lys substrate incubated for 30 mins by fluorometric activity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608555BDBM50608555(CHEMBL5269165)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608558BDBM50608558(CHEMBL5284956)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human recombinant HDAC1 using fluorogenic HDAC substrate measured after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 207629BDBM207629(US9265734, R01 | US9796664, Compound R01)
Affinity DataKi:  5nMAssay Description:Binding affinity to human recombinant HDAC3 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50510962BDBM50510962(CHEMBL4454646)
Affinity DataIC50: 5nMAssay Description:Inhibition of human HDAC3 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608558BDBM50608558(CHEMBL5284956)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of human HDAC3 using fluorogenic as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608558BDBM50608558(CHEMBL5284956)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of human recombinant HDAC3 using fluorogenic HDAC substrate measured after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608560BDBM50608560(CHEMBL5282899)
Affinity DataIC50: 6nMAssay Description:Inhibition of human HDAC1 by fluorescence based assay methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608556BDBM50608556(CHEMBL5281406)
Affinity DataIC50: 7nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608563BDBM50608563(CHEMBL5273740)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of human HDAC3 using fluorogenic as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608564BDBM50608564(CHEMBL5283088)
Affinity DataIC50: 9.70nMAssay Description:Inhibition of human HDAC using human HeLa cell nuclear extract measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470578BDBM50470578(CHEMBL4282111)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of human recombinant HDAC6 using Fluor-de-Lys as substrate at 50 uM for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608554BDBM50608554(CHEMBL5266056)
Affinity DataIC50: 12nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608563BDBM50608563(CHEMBL5273740)
Affinity DataIC50: 12nMAssay Description:Inhibition of human HDAC1 using fluorogenic as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608579BDBM50608579(CHEMBL5279294)
Affinity DataIC50: 13nMAssay Description:Inhibition of human HDAC3 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608577BDBM50608577(CHEMBL5281979)
Affinity DataIC50: 13nMAssay Description:Inhibition of HDAC6 (unknown origin) using Boc-Lys (Ac)-AMC as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608561BDBM50608561(CHEMBL5274036)
Affinity DataIC50: 14nMAssay Description:Inhibition of human HDAC using human HeLa cell nuclear extract measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608563BDBM50608563(CHEMBL5273740)
Affinity DataIC50: 14nMAssay Description:Inhibition of human HDAC using human HeLa cell nuclear extract measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608562BDBM50608562(CHEMBL5268468)
Affinity DataIC50: 16nMAssay Description:Inhibition of human HDAC using human HeLa cell nuclear extract measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50559735BDBM50559735(CHEMBL4740945)
Affinity DataIC50: 17nMAssay Description:Inhibition of human HDAC3 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608576BDBM50608576(CHEMBL5266011)
Affinity DataIC50: 17nMAssay Description:Inhibition of HDAC6 (unknown origin) using Boc-Lys (Ac)-AMC as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608561BDBM50608561(CHEMBL5274036)
Affinity DataIC50: 17nMAssay Description:Inhibition of human HDAC3 using fluorogenic as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50559742BDBM50559742(CHEMBL4741281)
Affinity DataIC50: 18nMAssay Description:Inhibition of human HDAC3 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 2(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50121210BDBM50121210(CHEMBL3622374)
Affinity DataIC50: 19nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 2(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608558BDBM50608558(CHEMBL5284956)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant HDAC2 using fluorogenic HDAC substrate measured after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470578BDBM50470578(CHEMBL4282111)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant HDAC3 using Fluor-de-Lys as substrate at 50 uM for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608562BDBM50608562(CHEMBL5268468)
Affinity DataIC50: 23nMAssay Description:Inhibition of human HDAC3 using fluorogenic as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50559731BDBM50559731(CHEMBL4779677)
Affinity DataIC50: 23nMAssay Description:Inhibition of human HDAC3 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608564BDBM50608564(CHEMBL5283088)
Affinity DataIC50: 24nMAssay Description:Inhibition of human HDAC3 using fluorogenic as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50559740BDBM50559740(CHEMBL4752047)
Affinity DataIC50: 24nMAssay Description:Inhibition of human HDAC3 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608564BDBM50608564(CHEMBL5283088)
Affinity DataIC50: 25nMAssay Description:Inhibition of human HDAC1 using fluorogenic as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608566BDBM50608566(CHEMBL5282033)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus by using Boc-L-Lys(Ac)-AMC as substrate measured after 24 hrs by fluorescence based an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608577BDBM50608577(CHEMBL5281979)
Affinity DataIC50: 27nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys (Ac)-AMC as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50559733BDBM50559733(CHEMBL4761763)
Affinity DataIC50: 28nMAssay Description:Inhibition of human HDAC3 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608561BDBM50608561(CHEMBL5274036)
Affinity DataIC50: 29nMAssay Description:Inhibition of human HDAC1 using fluorogenic as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254773BDBM50254773(CHEMBL3347696)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HDAC1 using (FAM)-labeled acetylated peptide substrate at 1 uM incubated for 17 hrs by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 2(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254773BDBM50254773(CHEMBL3347696)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HDAC2 using (FAM)-labeled acetylated peptide substrate at 1 uM incubated for 17 hrs by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470572BDBM50470572(CHEMBL4285537)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HDAC3More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254773BDBM50254773(CHEMBL3347696)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HDAC6 using (FAM)-labeled acetylated peptide substrate at 1 uM incubated for 17 hrs by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 8(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254773BDBM50254773(CHEMBL3347696)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HDAC8 using (FAM)-labeled acetylated peptide substrate at 1 uM incubated for 17 hrs by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608562BDBM50608562(CHEMBL5268468)
Affinity DataIC50: 31nMAssay Description:Inhibition of human HDAC1 using fluorogenic as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608579BDBM50608579(CHEMBL5279294)
Affinity DataIC50: 31nMAssay Description:Inhibition of human HDAC1 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608576BDBM50608576(CHEMBL5266011)
Affinity DataIC50: 32nMAssay Description:Inhibition of HDAC1 (unknown origin) using Boc-Lys (Ac)-AMC as substrate measured after 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608567BDBM50608567(CHEMBL5279348)
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant HDAC3 expressed in baculovirus by using Boc-L-Lys(Ac)-AMC as substrate measured after 24 hrs by fluorescence based an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608568BDBM50608568(CHEMBL5278816)
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant HDAC1 expressed in baculovirus by using Boc-L-Lys(Ac)-AMC as substrate measured after 24 hrs by fluorescence based an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50559734BDBM50559734(CHEMBL4749697)
Affinity DataIC50: 39nMAssay Description:Inhibition of human HDAC3 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50242041BDBM50242041(CHEMBL4103456)
Affinity DataIC50: 43nMAssay Description:Inhibition of HDAC3 (unknown origin) at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608567BDBM50608567(CHEMBL5279348)
Affinity DataIC50: 48nMAssay Description:Inhibition of human recombinant HDAC1 expressed in baculovirus by using Boc-L-Lys(Ac)-AMC as substrate measured after 24 hrs by fluorescence based an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPolyamine deacetylase HDAC10(Human)
Jadavpur University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50470578BDBM50470578(CHEMBL4282111)
Affinity DataIC50: 49nMAssay Description:Inhibition of human recombinant HDAC10 using Fluor-de-Lys as substrate at 50 uM for 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
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