Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50013277
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564261(CHEMBL4786031)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564254(CHEMBL4790137)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564255(CHEMBL4776328)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564273(CHEMBL4777182)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564261(CHEMBL4786031)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564264(CHEMBL4782066)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564271(CHEMBL4782988)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564257(CHEMBL4792567)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564263(CHEMBL4788954)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564259(CHEMBL4799886)
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564254(CHEMBL4790137)
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564265(CHEMBL4786350)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564260(CHEMBL4776974)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564258(CHEMBL4793650)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564273(CHEMBL4777182)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564265(CHEMBL4786350)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564258(CHEMBL4793650)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564255(CHEMBL4776328)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564259(CHEMBL4799886)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564265(CHEMBL4786350)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564263(CHEMBL4788954)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564256(CHEMBL4792980)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564256(CHEMBL4792980)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564254(CHEMBL4790137)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564257(CHEMBL4792567)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564256(CHEMBL4792980)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564264(CHEMBL4782066)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564255(CHEMBL4776328)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564263(CHEMBL4788954)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564262(CHEMBL4786063)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564260(CHEMBL4776974)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564261(CHEMBL4786031)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564266(CHEMBL4788942)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564271(CHEMBL4782988)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564258(CHEMBL4793650)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564266(CHEMBL4788942)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564262(CHEMBL4786063)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564266(CHEMBL4788942)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564259(CHEMBL4799886)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564264(CHEMBL4782066)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564257(CHEMBL4792567)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564273(CHEMBL4777182)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564262(CHEMBL4786063)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564274(CHEMBL4776599)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564260(CHEMBL4776974)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564274(CHEMBL4776599)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564274(CHEMBL4776599)
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564253(CHEMBL4782327)
Affinity DataIC50: 9.60nMAssay Description:Inhibition of recombinant human C-terminal His/FLAG-tagged HDAC1 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564253(CHEMBL4782327)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human full length C-terminal His-tagged HDAC8 expressed in sf9 insect cells using Boc-Lys(TFA)-AM as substrate incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Jiangsu Key Laboratory For Functional Substance of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50564253(CHEMBL4782327)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC2 (1 to end residues) expressed in sf9 insect cells using Boc-Lys(Ac)-AMC as substrate incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
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