Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50011142
TargetProteinase-activated receptor 1(Human)
Hebei University of Technology

Curated by ChEMBL
LigandPNGBDBM50545228(CHEMBL4639789)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Hebei University of Technology

Curated by ChEMBL
LigandPNGBDBM50261110(Ethyl [(3aR,4aR,8aR,9aS)-9(S)-[(E)-2-[5-(3-fluorop...)
Affinity DataIC50: 250nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Hebei University of Technology

Curated by ChEMBL
LigandPNGBDBM50545231(CHEMBL4632907)
Affinity DataIC50: 550nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Hebei University of Technology

Curated by ChEMBL
LigandPNGBDBM50545227(CHEMBL4633888)
Affinity DataIC50: 610nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Hebei University of Technology

Curated by ChEMBL
LigandPNGBDBM50545230(CHEMBL4639680)
Affinity DataIC50: 760nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Hebei University of Technology

Curated by ChEMBL
LigandPNGBDBM50545229(CHEMBL4633243)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed