Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50011816
Affinity DataKd: 1.90nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from recombinant human histamine H3 receptor stably transfected in HEK-293T cells membrane incubated for 9...More data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Agonist activity at human H3 receptor expressed in HEK293 cells preincubated for 30 mins followed by [35S]-GTPgammaS addition and measured after 30 m...More data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Agonist activity at human H3 receptor stably transfected in CHO-DUKX cells assessed as increase in cAMP accumulation by measuring reduction in forsko...More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human H3 receptor expressed in CHO cells assessed as increase in cAMP accumulation by measuring reduction in forskolin level incu...More data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Agonist activity at human H3 receptor expressed in CHO cells assessed as increase in cAMP accumulation by measuring reduction in forskolin level incu...More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from recombinant human histamine H3 receptor stably transfected in HEK-293T cells membrane incubated for 9...More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from recombinant human histamine H3 receptor stably transfected in HEK-293T cells membrane incubated for 9...More data for this Ligand-Target Pair
