Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50010712
LigandChemical structure of BindingDB Monomer ID 50541408BDBM50541408(CHEMBL4643140)
Affinity DataKi:  0.00400nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541406BDBM50541406(CHEMBL4649325)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541411BDBM50541411(CHEMBL4643006)
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of human CLR/RAMP1 by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 362044BDBM362044(US9833448, Example 4 | US10272077, Example 4)
Affinity DataKi:  0.0150nMAssay Description:Antagonist activity at human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541407BDBM50541407(CHEMBL4638635)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50184069BDBM50184069(CHEMBL207197 | N-((R)-1-((S)-6-amino-1-oxo-1-(4-(p...)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 391726BDBM391726(US10300056, Example 11 | N-[(2R)-3-(7-methyl-1H- |...)
Affinity DataKi:  0.0400nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541409BDBM50541409(CHEMBL4647045)
Affinity DataIC50: 0.0450nMAssay Description:Inhibition of human CLR/RAMP1 by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 361594BDBM361594(US9833448, Example 1 | US10272077, Example 1)
Affinity DataKi:  0.0670nMAssay Description:Antagonist activity at human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541405BDBM50541405(CHEMBL4633407)
Affinity DataKi:  0.110nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541412BDBM50541412(CHEMBL4644508)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541410BDBM50541410(CHEMBL4637301)
Affinity DataKi:  0.150nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541404BDBM50541404(CHEMBL4639133)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541413BDBM50541413(CHEMBL4649671)
Affinity DataKi:  0.25nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50047356BDBM50047356(CHEMBL3334624)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50224431BDBM50224431(N-[(3R,6S)-6-(2,3-difluorophenyl)-2-oxo-1-(2,2,2-t...)
Affinity DataKi:  0.770nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541403BDBM50541403(CHEMBL4641806)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50047357BDBM50047357(CHEMBL3334623)
Affinity DataIC50: 44nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541402BDBM50541402(CHEMBL4645875)
Affinity DataIC50: 250nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541401BDBM50541401(CHEMBL4634626)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50541400BDBM50541400(CHEMBL4634646)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50173483BDBM50173483((S)-6-Amino-2-[(R)-3-(3,5-dibromo-4-hydroxy-phenyl...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed