Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50009312
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527071BDBM50527071(CHEMBL4514624)
Affinity DataKi:  1.30nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453611BDBM50453611(CHEMBL4207081)
Affinity DataKi:  11nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527063BDBM50527063(CHEMBL4534285)
Affinity DataKi:  11nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453612BDBM50453612(CHEMBL4216774)
Affinity DataKi:  17nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527071BDBM50527071(CHEMBL4514624)
Affinity DataKi:  18nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453611BDBM50453611(CHEMBL4207081)
Affinity DataKi:  19nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50453612BDBM50453612(CHEMBL4216774)
Affinity DataKi:  27nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 3(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527068BDBM50527068(CHEMBL468766 | CHEBI:17734)
Affinity DataIC50: 90nMAssay Description:Inhibition of human SERCA3a expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527068BDBM50527068(CHEMBL468766 | CHEBI:17734)
Affinity DataIC50: 90nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527068BDBM50527068(CHEMBL468766 | CHEBI:17734)
Affinity DataIC50: 90nMAssay Description:Inhibition of rabbit SERCA1b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527063BDBM50527063(CHEMBL4534285)
Affinity DataIC50: 210nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527063BDBM50527063(CHEMBL4534285)
Affinity DataIC50: 210nMAssay Description:Inhibition of rabbit SERCA1b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 3(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527063BDBM50527063(CHEMBL4534285)
Affinity DataIC50: 210nMAssay Description:Inhibition of human SERCA3a expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527076BDBM50527076(CHEMBL4436782)
Affinity DataIC50: 270nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410532BDBM50410532(4-NONYLPHENOL)
Affinity DataIC50: 350nMAssay Description:Inhibition of SERCA1a in rabbit microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 3(Mouse)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410532BDBM50410532(4-NONYLPHENOL)
Affinity DataIC50: 350nMAssay Description:Inhibition of SERCA3 in mouse testicular microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410532BDBM50410532(4-NONYLPHENOL)
Affinity DataIC50: 350nMAssay Description:Inhibition of rabbit SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410532BDBM50410532(4-NONYLPHENOL)
Affinity DataIC50: 350nMAssay Description:Inhibition of SERCA2b in mouse testicular microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50150793BDBM50150793(4,4'-(propane-2,2-diyl)bis(2,6-dibromophenol) | 3,...)
Affinity DataIC50: 500nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50323389BDBM50323389(Calmidazolium | CHEMBL1208858)
Affinity DataIC50: 500nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a incubated for 10 mins by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527067BDBM50527067(CHEMBL4531692)
Affinity DataIC50: 610nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527070BDBM50527070(CHEMBL4467779)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25524BDBM25524(CHEMBL13045 | 17,18-dimethoxy-21-methyl-5,7-dioxa-...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a incubated for 10 mins by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527074BDBM50527074(CHEMBL4536029)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a by malachite green based colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 3(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 176764BDBM176764(US9688816, 7 | 2,5-Di-tert-butylhydroquinone | CAS...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human SERCA3a expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 29608BDBM29608(Diphenylolpropane | Bisphenol A (BPA) | US9688816,...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 176764BDBM176764(US9688816, 7 | 2,5-Di-tert-butylhydroquinone | CAS...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rabbit SERCA1b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Rat)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 29608BDBM29608(Diphenylolpropane | Bisphenol A (BPA) | US9688816,...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat cerebellar microsomes SERCA2b by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 176764BDBM176764(US9688816, 7 | 2,5-Di-tert-butylhydroquinone | CAS...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140172BDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 3(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50854BDBM50854(MLS000028812 | SMR000058863 | PAXILLINE | cid_1050...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of SERCA3 in human platelet microsomes by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50854BDBM50854(MLS000028812 | SMR000058863 | PAXILLINE | cid_1050...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of SERCA2b in human platelet microsomes by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50854BDBM50854(MLS000028812 | SMR000058863 | PAXILLINE | cid_1050...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Pig)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31774BDBM31774(cid_2812 | CHEMBL104 | Canesten | Mycelex | Lotrim...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of pig gastric mucosa Potassium-transporting ATPase by malachite green based colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140172BDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of rabbit SERCA1b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50187657BDBM50187657(3,6-dihydroxy-flavone | 3,6-dihydroxy-2-phenyl-4H-...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a preincubated for 10 mins followed by addition of ATP and measured after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50139422BDBM50139422(CHEMBL1495071)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 3(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140172BDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of SERCA3 in human platelet microsomes by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140172BDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of SERCA2b in human platelet microsomes by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527072BDBM50527072(CHEMBL524065)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a by malachite green based colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 3(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140172BDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataKi:  8.60E+3nMAssay Description:Inhibition of human SERCA3a expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50049391BDBM50049391(norizalpinin | 3,5,7-trihydroxy-2-phenyl-4H-benzop...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a preincubated for 10 mins followed by addition of ATP and measured after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 7460BDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a preincubated for 10 mins followed by addition of ATP and measured after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070942BDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50297393BDBM50297393(Ethyl 2-Amino-6-(3',5'-dimethoxyphenyl)-4-(2-ethox...)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20625BDBM20625(CHEMBL411 | Stilbestrol | 4-[(3E)-4-(4-hydroxyphen...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of rabbit microsomes SERCA1a by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 78433BDBM78433(2-[4-[3-[2-(trifluoromethyl)phenothiazin-10-yl]pro...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a incubated for 10 mins by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409816BDBM50409816(ABAMECTIN)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of rabbit SERCA1a preincubated for 10 mins followed by addition of ATP and measured after 10 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50527075BDBM50527075(CHEMBL4592594)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rabbit SERCA1a incubated for 10 mins by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001888BDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of rabbit skeletal muscle microsomes SERCA1a incubated for 10 mins by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
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