Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50007645
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511159BDBM50511159(CHEMBL4550946)
Affinity DataIC50: 13nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511162BDBM50511162(CHEMBL4575812)
Affinity DataIC50: 14nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511154BDBM50511154(CHEMBL4442374)
Affinity DataIC50: 19nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511152BDBM50511152(CHEMBL4474836)
Affinity DataIC50: 25nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 100152BDBM100152(cid_5359389 | SMR001233259 | HARMINE | 7-methoxy-1...)
Affinity DataIC50: 27nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511155BDBM50511155(CHEMBL4456985)
Affinity DataIC50: 27nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511150BDBM50511150(CHEMBL4440790)
Affinity DataIC50: 39nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511164BDBM50511164(CHEMBL4514653)
Affinity DataIC50: 56nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511156BDBM50511156(CHEMBL4521356)
Affinity DataIC50: 64nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511161BDBM50511161(CHEMBL4579529)
Affinity DataIC50: 74nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511165BDBM50511165(CHEMBL4563765)
Affinity DataIC50: 84nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511158BDBM50511158(CHEMBL4437998)
Affinity DataIC50: 97nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511157BDBM50511157(CHEMBL4552025)
Affinity DataIC50: 98nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511160BDBM50511160(CHEMBL4513287)
Affinity DataIC50: 112nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511153BDBM50511153(CHEMBL4564623)
Affinity DataIC50: 139nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50379523BDBM50379523(CHEMBL2012558)
Affinity DataIC50: 152nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511151BDBM50511151(CHEMBL4483653)
Affinity DataIC50: 168nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511147BDBM50511147(CHEMBL4476003)
Affinity DataIC50: 168nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511149BDBM50511149(CHEMBL4438785)
Affinity DataIC50: 215nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511148BDBM50511148(CHEMBL4539999)
Affinity DataIC50: 950nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50511163BDBM50511163(CHEMBL4528315)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed