Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50007973
TargetT-type calcium channel alpha 1G subunit(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514579(CHEMBL4575063)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at mouse Cav3.1 expressed in HEK293T cells assessed as increase in current amplitude at holding potential of -100 mV by whole cell e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514580(CHEMBL4455355)
Affinity DataEC50:  1.25E+4nMAssay Description:Agonist activity at Cav3.1 (unknown origin) expressed in HEK293T cells assessed as increase in current amplitude at holding potential of -100 mV by w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetT-type calcium channel alpha 1G subunit(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514577(CHEMBL3581591)
Affinity DataIC50: 190nMAssay Description:Antagonist activity at mouse Cav3.1 expressed in HEK293T cells assessed as inhibition of current amplitude at holding potential of -100 mV by whole c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetT-type calcium channel alpha 1G subunit(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50514578(CHEMBL4464354)
Affinity DataIC50: 2.30E+3nMAssay Description:Antagonist activity at mouse Cav3.1 expressed in HEK293T cells assessed as inhibition of current amplitude at holding potential of -100 mV by whole c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetT-type calcium channel alpha 1G subunit(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50090184(CHEMBL3581573)
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at mouse Cav3.1 expressed in HEK293T cells assessed as inhibition of current amplitude at holding potential of -100 mV by whole c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed