Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50010678
TargetGlucose-dependent insulinotropic receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50013909(CHEMBL3260505)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at GPR119 (unknown origin) assessed as increase in cAMP level by cAMP HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50541160(CHEMBL4648870)
Affinity DataEC50:  4.90nMAssay Description:Agonist activity at GPR119 (unknown origin) assessed as increase in cAMP level by cAMP HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50541161(CHEMBL4647675)
Affinity DataEC50:  8.80nMAssay Description:Agonist activity at GPR119 (unknown origin) assessed as increase in cAMP level by cAMP HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50541162(CHEMBL4641634)
Affinity DataEC50:  10nMAssay Description:Agonist activity at GPR119 (unknown origin) assessed as increase in cAMP level by cAMP HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50541159(CHEMBL4639029)
Affinity DataEC50:  71nMAssay Description:Agonist activity at GPR119 (unknown origin) assessed as increase in cAMP level by cAMP HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50541158(CHEMBL4645561)
Affinity DataEC50:  107nMAssay Description:Agonist activity at GPR119 (unknown origin) assessed as increase in cAMP level by cAMP HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50541157(CHEMBL4648982)
Affinity DataEC50:  108nMAssay Description:Agonist activity at GPR119 (unknown origin) assessed as increase in cAMP level by cAMP HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50541156(CHEMBL4637425)
Affinity DataEC50:  113nMAssay Description:Agonist activity at GPR119 (unknown origin) assessed as increase in cAMP level by cAMP HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50541155(CHEMBL4645380)
Affinity DataEC50:  678nMAssay Description:Agonist activity at GPR119 (unknown origin) assessed as increase in cAMP level by cAMP HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM29080(Oleamide MEA | Oleoyl monoethanolamide | CHEMBL280...)
Affinity DataEC50:  930nMAssay Description:Agonist activity at GPR119 (unknown origin) assessed as increase in cAMP level by cAMP HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed