Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50010485
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 257nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 283nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 299nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.99E+3nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetCholinesterase(Horse)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 7.05E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 7.92E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.86E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 9.45E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.94E+4nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.16E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.22E+4nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.66E+4nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electric eel)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins by...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.59E+4nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetCholinesterase(Horse)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 7.25E+4nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 7.54E+4nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.25E+4nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.37E+4nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.04E+5nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetCholinesterase(Horse)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins ...More data for this Ligand-Target Pair
TargetCholinesterase(Horse)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.34E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.41E+5nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetCholinesterase(Horse)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.49E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins ...More data for this Ligand-Target Pair
TargetCholinesterase(Horse)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.88E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.89E+5nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetCholinesterase(Horse)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.08E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.93E+5nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rat)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of MAO-B in Wistar rat liver using 4-trifluoromethyl benzylamine as substrate preincubated for 20 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetCholinesterase(Horse)
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
University of Jinan-Shandong Academy of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of equine serum BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition measured after 20 mins ...More data for this Ligand-Target Pair
