Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50007103
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506303(CHEMBL4546597)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506307(CHEMBL4541779)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506296(CHEMBL4537162)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in CHOK1 cells assessed as increase in cAMP level measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506305(CHEMBL4456573)
Affinity DataEC50:  65nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506296(CHEMBL4537162)
Affinity DataEC50:  193nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506304(CHEMBL4560445)
Affinity DataEC50:  831nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506306(CHEMBL4460622)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506296(CHEMBL4537162)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at recombinant human V1a receptor expressed in CHO cells by calcium no wash plus assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506298(CHEMBL4442222)
Affinity DataEC50:  57nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506302(CHEMBL4546106)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506305(CHEMBL4456573)
Affinity DataEC50:  464nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506296(CHEMBL4537162)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506296(CHEMBL4537162)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at recombinant human V1b receptor expressed in RBL cells by calcium no wash plus assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506304(CHEMBL4560445)
Affinity DataEC50:  52nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506303(CHEMBL4546597)
Affinity DataEC50:  173nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506302(CHEMBL4546106)
Affinity DataEC50:  19nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506301(CHEMBL4532581)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506300(CHEMBL4589487)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506299(CHEMBL4550811)
Affinity DataEC50:  14nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  3nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506298(CHEMBL4442222)
Affinity DataEC50:  10nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Calibr At The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50506297(CHEMBL4463103)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at recombinant human Gi/Go-coupled OTR expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment measured after 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed