Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50008517
TargetAdenosine receptor A1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50520046(CHEMBL1340426)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1A receptor expressed in human CHO cell membranes incubated for 60 mins by scintillation counting met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50520046(CHEMBL1340426)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50520047(CHEMBL1465169)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50520044(CHEMBL1406529)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50520044(CHEMBL1406529)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50520045(CHEMBL1712711)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1A receptor expressed in human CHO cell membranes incubated for 60 mins by scintillation counting met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50520045(CHEMBL1712711)
Affinity DataKi:  4.90E+3nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50520047(CHEMBL1465169)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed