Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50007074
TargetAryl hydrocarbon receptor(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50506038(CHEMBL4580482)
Affinity DataEC50:  49nMAssay Description:Binding affinity to AhR (unknown origin) relative to TCDDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Mouse)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50506039(CHEMBL1324296 | US11891386, Compound 002)
Affinity DataKd:  3nMAssay Description:Displacement of [3H]TCDD from mouse AhRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50028963(beta-naphthoflavone | 3-phenyl-1H-benzo[f]chromen-...)
Affinity DataEC50:  8.40nMAssay Description:Agonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50506038(CHEMBL4580482)
Affinity DataKd:  0.130nMAssay Description:Binding affinity to AhR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Mouse)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50239186(CHEBI:50182 | 1,1-Bis(3''-Indolyl)Methane | 3,3''-...)
Affinity DataEC50:  7.80E+4nMAssay Description:Displacement of 2-azido-3-[125I]7,8-dibromodibenzo-pdioxin from C57BL/6J mouse liver AhR relative to TCDDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Mouse)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50239186(CHEBI:50182 | 1,1-Bis(3''-Indolyl)Methane | 3,3''-...)
Affinity DataKd:  90nMAssay Description:Displacement of 2-azido-3-[125I]7,8-dibromodibenzo-pdioxin from C57BL/6J mouse liver AhRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50506040(CHEMBL4536502)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H] 3-MC from AhR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Mouse)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50439845(CHEMBL2420083)
Affinity DataIC50: 21nMAssay Description:Displacement of 2-azido-3-[125I]7,8-dibromodibenzo-pdioxin from C57BL/6J mouse liver AhR incubated for 20 mins by gamma counting based autoradiograph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Mouse)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50014323(CHEMBL283196 | alpha-naphthoflavone | 2-PHENYL-4H-...)
Affinity DataIC50: 25nMAssay Description:Displacement of 2-azido-3-[125I]7,8-dibromodibenzo-pdioxin from C57BL/6J mouse liver AhR incubated for 20 mins by gamma counting based autoradiograph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Human)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50506041(CHEBI:16946 | L-kynurenine)
Affinity DataKi:  2.16E+4nMAssay Description:Inhibition of AhR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed