Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50007071
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50455084(CHEMBL4214098)
Affinity DataIC50: 2.45E+3nMAssay Description:Inhibition of human NNMT using nicotinamide as substrate preincubated for 30 mins followed by substrate addition in presence of AdoMet and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAdenosylhomocysteinase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of SAHH (unknown origin) using SAH as substrate preincubated for 10 mins followed by susbtrate addition by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of NTMT1 (unknown origin) using GPKRIA peptide as substrate preincubated for 10 mins in presence of AdoMet followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant rat His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using H4-21 peptide as susbtrate preincubated for 10 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human His-tagged SETD7 (1 to 366 residues) expressed in Escherichia coli using H3-21 peptide as susbtrate preincubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human G9a (913 to 1193 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using H3-21 peptide preincubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N- terminal His6 tagged human INMT expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL using tryptamine as substrate preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-terminal His6 tagged PNMT using norepinephrine as substrate preincubated for 10 mins in presence of AdoMet followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataKi:  1.60nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataKi:  1.90nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataKi:  1.90nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataKi:  2.60nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506000(CHEMBL4445337)
Affinity DataKi:  6.80nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506009(CHEMBL4476197)
Affinity DataKi:  16nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506011(CHEMBL4436698)
Affinity DataKi:  43nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506015(CHEMBL4556842)
Affinity DataKi:  51nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506008(CHEMBL4439305)
Affinity DataKi:  52nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506003(CHEMBL4522203)
Affinity DataKi:  150nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506002(CHEMBL4437502)
Affinity DataKi:  540nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506013(CHEMBL4557645)
Affinity DataKi:  840nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506005(CHEMBL4517536)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506010(CHEMBL4467665)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506004(CHEMBL4542138)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506006(CHEMBL4454317)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50247635(CHEMBL4100002)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506001(CHEMBL4581026)
Affinity DataKi:  1.18E+4nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506014(CHEMBL4458772)
Affinity DataKi:  2.73E+4nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506007(CHEMBL4572902)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50506012(CHEMBL4561228)
Affinity DataKi:  3.33E+4nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNicotinamide N-methyltransferase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50106187(Benzoylamide | Benzenecarboxamide | CHEMBL267373 |...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of full-length human N-terminal TEV cleavage site NNMT (1 to 270 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIPL cells us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed