Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50008444
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50103521(CHEBI:8228 | Actos | Duetact | Pioglitazone | US20...)
Affinity DataEC50:  1.40E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma transfected in COS7 cells co-transfected with pGAL5-TK-pGL3 and pRennilla-CMV incubated for 39 hrs by d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50043280(4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimi...)
Affinity DataEC50:  4.28E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma transfected in COS7 cells co-transfected with pGAL5-TK-pGL3 and pRennilla-CMV incubated for 39 hrs by d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50324039(4'-[(2-Propyl-1H-benzo[d]imidazol-1-yl)methyl]biph...)
Affinity DataEC50:  7.22E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma transfected in COS7 cells co-transfected with pGAL5-TK-pGL3 and pRennilla-CMV incubated for 39 hrs by d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50519389(CHEMBL4587597)
Affinity DataEC50:  8.25E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma transfected in COS7 cells co-transfected with pGAL5-TK-pGL3 and pRennilla-CMV incubated for 39 hrs by d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50519387(CHEMBL4435043)
Affinity DataEC50:  8.66E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma transfected in COS7 cells co-transfected with pGAL5-TK-pGL3 and pRennilla-CMV incubated for 39 hrs by d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50519390(CHEMBL4552317)
Affinity DataEC50:  8.67E+3nMAssay Description:Transactivation of Gal4-fused human PPARgamma transfected in COS7 cells co-transfected with pGAL5-TK-pGL3 and pRennilla-CMV incubated for 39 hrs by d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50519386(CHEMBL4466036)
Affinity DataEC50:  1.11E+4nMAssay Description:Transactivation of Gal4-fused human PPARgamma transfected in COS7 cells co-transfected with pGAL5-TK-pGL3 and pRennilla-CMV incubated for 39 hrs by d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50519388(CHEMBL4538895)
Affinity DataEC50:  1.21E+4nMAssay Description:Transactivation of Gal4-fused human PPARgamma transfected in COS7 cells co-transfected with pGAL5-TK-pGL3 and pRennilla-CMV incubated for 39 hrs by d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed