Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50007033
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505559(CHEMBL4441303)
Affinity DataIC50: 0.0940nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505555(CHEMBL4447348)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50033762(Gallinamide A)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505557(CHEMBL4527930)
Affinity DataIC50: 0.470nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505568(CHEMBL4482954)
Affinity DataIC50: 0.490nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505555(CHEMBL4447348)
Affinity DataIC50: 0.632nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505562(CHEMBL4445744)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505554(CHEMBL4564747)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505557(CHEMBL4527930)
Affinity DataIC50: 0.790nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505563(CHEMBL4527329)
Affinity DataIC50: 0.840nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505566(CHEMBL4582558)
Affinity DataIC50: 1nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505565(CHEMBL4474668)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505559(CHEMBL4441303)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505561(CHEMBL4475810)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505564(CHEMBL4527867)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505560(CHEMBL4471760)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505562(CHEMBL4445744)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505560(CHEMBL4471760)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505568(CHEMBL4482954)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505565(CHEMBL4474668)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505567(CHEMBL4457500)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505564(CHEMBL4527867)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505561(CHEMBL4475810)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505563(CHEMBL4527329)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505566(CHEMBL4582558)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505554(CHEMBL4564747)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50033762(Gallinamide A)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50033762(Gallinamide A)
Affinity DataIC50: 5nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505567(CHEMBL4457500)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505558(CHEMBL4514842)
Affinity DataIC50: 37nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505558(CHEMBL4514842)
Affinity DataIC50: 77nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCruzipain(Trypanosoma cruzi)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505556(CHEMBL4468530)
Affinity DataIC50: 81nMAssay Description:Inhibition of recombinant Trypanosoma cruzi Cruzain expressed in Pichia pastoris using Z-Phe-Arg-AMC substrate incubated for 30 mins by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProcathepsin L(Human)
The University of Jordan

Curated by ChEMBL
LigandPNGBDBM50505556(CHEMBL4468530)
Affinity DataIC50: 376nMAssay Description:Inhibition of human cathepsin L using fluorogenic substrate cbz-FR-AMC monitored for 90 to 120 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed