Compile Data Set for Download or QSAR
Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 50009443
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528930(CHEMBL4471658)
Affinity DataIC50: 0.890nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528926(CHEMBL4565200)
Affinity DataIC50: 26nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528924(CHEMBL4473519)
Affinity DataIC50: 58nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528925(CHEMBL4540218)
Affinity DataIC50: 62nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528932(CHEMBL4554053)
Affinity DataIC50: 94nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528930(CHEMBL4471658)
Affinity DataIC50: 100nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528930(CHEMBL4471658)
Affinity DataIC50: 100nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataIC50: 110nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528931(CHEMBL4520982)
Affinity DataIC50: 175nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528933(CHEMBL4449756)
Affinity DataIC50: 195nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528926(CHEMBL4565200)
Affinity DataIC50: 280nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528926(CHEMBL4565200)
Affinity DataIC50: 282nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528928(CHEMBL4520184)
Affinity DataIC50: 757nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528927(CHEMBL4517296)
Affinity DataIC50: 791nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528925(CHEMBL4540218)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528925(CHEMBL4540218)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528929(CHEMBL4446507)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528932(CHEMBL4554053)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528932(CHEMBL4554053)
Affinity DataIC50: 3.55E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528924(CHEMBL4473519)
Affinity DataIC50: 5.25E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528924(CHEMBL4473519)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528927(CHEMBL4517296)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528927(CHEMBL4517296)
Affinity DataIC50: 6.46E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50131925(N-(4-(4-(2,4-dichlorophenyl)piperazin-1-yl)butyl)-...)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]-7-OH-DPAT from rat brain membrane D3 receptor expressed in Sf9 cells incubated for 60 mins by liquid scintillation counting meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528930(CHEMBL4471658)
Affinity DataKi:  0.230nMAssay Description:Inhibition of FAAH in mouse brain membranes assessed as inhibitory constant using [14C]-AEA as substrate incubated for 15 mins by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528926(CHEMBL4565200)
Affinity DataKi:  6.90nMAssay Description:Inhibition of FAAH in mouse brain membranes assessed as inhibitory constant using [14C]-AEA as substrate incubated for 15 mins by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528924(CHEMBL4473519)
Affinity DataKi:  16nMAssay Description:Inhibition of FAAH in mouse brain membranes assessed as inhibitory constant using [14C]-AEA as substrate incubated for 15 mins by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528925(CHEMBL4540218)
Affinity DataKi:  16nMAssay Description:Inhibition of FAAH in mouse brain membranes assessed as inhibitory constant using [14C]-AEA as substrate incubated for 15 mins by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528925(CHEMBL4540218)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528925(CHEMBL4540218)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528932(CHEMBL4554053)
Affinity DataKi:  25nMAssay Description:Inhibition of FAAH in mouse brain membranes assessed as inhibitory constant using [14C]-AEA as substrate incubated for 15 mins by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528925(CHEMBL4540218)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528925(CHEMBL4540218)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528932(CHEMBL4554053)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528932(CHEMBL4554053)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528931(CHEMBL4520982)
Affinity DataKi:  46nMAssay Description:Inhibition of FAAH in mouse brain membranes assessed as inhibitory constant using [14C]-AEA as substrate incubated for 15 mins by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528933(CHEMBL4449756)
Affinity DataKi:  50nMAssay Description:Inhibition of FAAH in mouse brain membranes assessed as inhibitory constant using [14C]-AEA as substrate incubated for 15 mins by scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528927(CHEMBL4517296)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528927(CHEMBL4517296)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528932(CHEMBL4554053)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528932(CHEMBL4554053)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528927(CHEMBL4517296)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528927(CHEMBL4517296)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528924(CHEMBL4473519)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528930(CHEMBL4471658)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528924(CHEMBL4473519)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528930(CHEMBL4471658)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528930(CHEMBL4471658)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528930(CHEMBL4471658)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50528926(CHEMBL4565200)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
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