Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50009437
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528877(CHEMBL4450162)
Affinity DataEC50:  9.62E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50130918(CHEMBL3632943)
Affinity DataEC50:  1.21E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50130902(CHEMBL3632949)
Affinity DataEC50:  1.04E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528882(CHEMBL4448642)
Affinity DataEC50:  2.03E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528881(CHEMBL4448581)
Affinity DataEC50:  2.58E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50130894(CHEMBL3632627)
Affinity DataEC50:  3.03E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528880(CHEMBL4518138)
Affinity DataEC50:  2.97E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528879(CHEMBL4441750)
Affinity DataEC50:  2.03E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528878(CHEMBL4436181)
Affinity DataEC50:  3.01E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528883(CHEMBL4557359)
Affinity DataEC50:  1.26E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528876(CHEMBL4466082)
Affinity DataEC50:  4.69E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528875(CHEMBL4441683)
Affinity DataEC50:  6.66E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528874(CHEMBL4566536)
Affinity DataEC50:  120nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528873(CHEMBL4447851)
Affinity DataEC50:  2.30E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528872(CHEMBL3121587)
Affinity DataEC50:  3.42E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528871(CHEMBL4467008)
Affinity DataEC50:  2.45E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528870(CHEMBL4447216)
Affinity DataEC50:  5.55E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528869(CHEMBL4437194)
Affinity DataEC50:  3.34E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528889(CHEMBL4515076)
Affinity DataEC50:  1.19E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528895(CHEMBL4449675)
Affinity DataEC50:  8.80E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50130912(CHEMBL3632957)
Affinity DataEC50:  4.74E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528894(CHEMBL4442830)
Affinity DataEC50:  2.23E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528893(CHEMBL4441811)
Affinity DataEC50:  2.10E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528892(CHEMBL4571467)
Affinity DataEC50:  7.32E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528891(CHEMBL4448140)
Affinity DataEC50:  2.02E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50130916(CHEMBL3632945)
Affinity DataEC50:  4.07E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528890(CHEMBL4578763)
Affinity DataEC50:  1.33E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528868(CHEMBL4540228)
Affinity DataEC50:  1.75E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50130919(CHEMBL3632942)
Affinity DataEC50:  2.40E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528888(CHEMBL4535717)
Affinity DataEC50:  3.57E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528887(CHEMBL3121589)
Affinity DataEC50:  1.51E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50130913(CHEMBL3632958)
Affinity DataEC50:  1.33E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528886(CHEMBL4456858)
Affinity DataEC50:  1.67E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528885(CHEMBL4448855)
Affinity DataEC50:  1.76E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528884(CHEMBL4560147)
Affinity DataEC50:  4.70E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528851(CHEMBL4475517)
Affinity DataEC50:  1.64E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528858(CHEMBL4455067)
Affinity DataEC50:  6.00E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528857(CHEMBL4519986)
Affinity DataEC50:  8.90E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50130908(CHEMBL3632954)
Affinity DataEC50:  3.36E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528856(CHEMBL4471852)
Affinity DataEC50:  90nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528855(CHEMBL4458677)
Affinity DataEC50:  2.52E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528854(CHEMBL4483791)
Affinity DataEC50:  1.44E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528853(CHEMBL4474400)
Affinity DataEC50:  1.21E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528852(CHEMBL4473940)
Affinity DataEC50:  1.10E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50130907(ALISOL A)
Affinity DataEC50:  1.02E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528850(CHEMBL4466386)
Affinity DataEC50:  5.60E+3nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528849(CHEMBL4437372)
Affinity DataEC50:  1.02E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528848(CHEMBL4536937)
Affinity DataEC50:  290nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50528847(CHEMBL4577420)
Affinity DataEC50:  110nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50130900(CHEMBL3632947)
Affinity DataEC50:  6.49E+4nMAssay Description:Transactivation of FXR (unknown origin) transfected in HepG2 cells co-expressing pBSEP/pGL4.74 incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
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