Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50009162
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525859(CHEMBL4467539)
Affinity DataIC50: 550nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525858(CHEMBL4483375)
Affinity DataIC50: 850nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525856(CHEMBL4447887)
Affinity DataIC50: 1.04E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525857(CHEMBL4558377)
Affinity DataIC50: 1.26E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataIC50: 1.32E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525853(CHEMBL4473613)
Affinity DataIC50: 1.56E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525854(CHEMBL4538661)
Affinity DataIC50: 2.08E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525851(CHEMBL4443680)
Affinity DataIC50: 2.21E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525862(CHEMBL4438851)
Affinity DataIC50: 2.56E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525861(CHEMBL4562339)
Affinity DataIC50: 3.02E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525852(CHEMBL4459595)
Affinity DataIC50: 3.54E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525850(CHEMBL4450139)
Affinity DataIC50: 3.72E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525855(CHEMBL4564123)
Affinity DataIC50: 3.87E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Luoyang Normal University

Curated by ChEMBL
LigandPNGBDBM50525860(CHEMBL4519947)
Affinity DataIC50: 3.94E+3nMAssay Description:Displacement of fluormone-AL Green from His-tagged/GST-fused recombinant rat androgen receptor LBD expressed in insect cells measured after 4 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed