Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50009614
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50000541(Leutrol | CHEMBL93 | N-(1-Benzo(b)thien-2-ylethyl)...)
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human 5-lipoxygenase expressed in Escherichia coli BL21 (DE3) cells using arachidonic acid as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50000541(Leutrol | CHEMBL93 | N-(1-Benzo(b)thien-2-ylethyl)...)
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human 5-lipoxygenase expressed in Escherichia coli BL21 (DE3) cells using arachidonic acid as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530488(CHEMBL4527956)
Affinity DataIC50: 900nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530488(CHEMBL4527956)
Affinity DataIC50: 900nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530484(CHEMBL4454636)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530484(CHEMBL4454636)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530492(CHEMBL522025 | CHEBI:7061)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530492(CHEMBL522025 | CHEBI:7061)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530489(CHEMBL4561848)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530489(CHEMBL4561848)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM179805(Myxochelin A)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM179805(Myxochelin A)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530485(CHEMBL4464140)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530485(CHEMBL4464140)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530491(CHEMBL4586522)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530491(CHEMBL4586522)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530486(CHEMBL4522098)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530486(CHEMBL4522098)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530494(CHEMBL4438375)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530494(CHEMBL4438375)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530490(CHEMBL4546578)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530483(CHEMBL4474339)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530487(CHEMBL4445605)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530493(CHEMBL4476763)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530493(CHEMBL4476763)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530483(CHEMBL4474339)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530490(CHEMBL4546578)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
Institute For Natural Product Research and Infection Biology

Curated by ChEMBL
LigandPNGBDBM50530487(CHEMBL4445605)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human 5-lipoxygenase using arachidonic acid as substrate preincubated for 10 mins followed by susbtrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed