Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50008768
TargetHistone-lysine N-methyltransferase SETDB1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50521986(CHEMBL4451286)
Affinity DataKd:  1.00E+7nMAssay Description:Binding affinity to N-terminally biotinylated human SETDB1 Tudor domain (197 to 403 residues) expressed in Escherichia coli BL21(DE3)-pRARE2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase SETDB1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50521987(CHEMBL4542222)
Affinity DataKd:  2.70E+6nMAssay Description:Binding affinity to N-terminally biotinylated human SETDB1 Tudor domain (197 to 403 residues) expressed in Escherichia coli BL21(DE3)-pRARE2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase SETDB1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50521988(CHEMBL4456448)
Affinity DataKd:  1.27E+6nMAssay Description:Binding affinity to N-terminally biotinylated human SETDB1 Tudor domain (197 to 403 residues) expressed in Escherichia coli BL21(DE3)-pRARE2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase SETDB1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50521989(CHEMBL4453131)
Affinity DataKd:  4.00E+6nMAssay Description:Binding affinity to N-terminally biotinylated human SETDB1 Tudor domain (197 to 403 residues) expressed in Escherichia coli BL21(DE3)-pRARE2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase SETDB1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50521990(CHEMBL4576037)
Affinity DataKd:  3.50E+6nMAssay Description:Binding affinity to N-terminal His6-tagged human SETDB1 Tudor domain (197 to 403 residues) expressed in Escherichia coli BL21(DE3)-pRARE2 cells by IT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase SETDB1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50521990(CHEMBL4576037)
Affinity DataKd:  3.50E+6nMAssay Description:Binding affinity to N-terminally biotinylated human SETDB1 Tudor domain (197 to 403 residues) expressed in Escherichia coli BL21(DE3)-pRARE2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase SETDB1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50521991(CHEMBL4589361)
Affinity DataKd:  7.70E+6nMAssay Description:Binding affinity to N-terminally biotinylated human SETDB1 Tudor domain (197 to 403 residues) expressed in Escherichia coli BL21(DE3)-pRARE2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase SETDB1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50521992(CHEMBL4455427)
Affinity DataKd:  2.50E+6nMAssay Description:Binding affinity to N-terminally biotinylated human SETDB1 Tudor domain (197 to 403 residues) expressed in Escherichia coli BL21(DE3)-pRARE2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase SETDB1(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50521989(CHEMBL4453131)
Affinity DataKd:  4.00E+6nMAssay Description:Binding affinity to N-terminal His6-tagged human SETDB1 Tudor domain (197 to 403 residues) expressed in Escherichia coli BL21(DE3)-pRARE2 cells by IT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed