Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50008062
TargetHistone deacetylase 6(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant HDAC6 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 61nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 3(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 62nMAssay Description:Inhibition of recombinant HDAC3 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515347(CHEMBL4461759)
Affinity DataIC50: 160nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 173nMAssay Description:Inhibition of recombinant HDAC2 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515343(CHEMBL4515273)
Affinity DataIC50: 190nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515350(CHEMBL4452725)
Affinity DataIC50: 200nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515353(CHEMBL4449504)
Affinity DataIC50: 230nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50346552(CHEMBL1797936)
Affinity DataIC50: 230nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515362(CHEMBL4436898)
Affinity DataIC50: 290nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50346552(CHEMBL1797936)
Affinity DataIC50: 400nMAssay Description:Inhibition of p300 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515367(CHEMBL4448489)
Affinity DataIC50: 470nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515354(CHEMBL4452893)
Affinity DataIC50: 560nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515368(CHEMBL4474848)
Affinity DataIC50: 580nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515349(CHEMBL4526489)
Affinity DataIC50: 670nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515369(CHEMBL4449804)
Affinity DataIC50: 860nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515351(CHEMBL4443388)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515365(CHEMBL4564246)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515366(CHEMBL4515579)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515344(CHEMBL4466615)
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515372(CHEMBL4537592)
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515345(CHEMBL4560819)
Affinity DataIC50: 3.73E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515348(CHEMBL4535402)
Affinity DataIC50: 4.06E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of recombinant HDAC8 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515363(CHEMBL4578596)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515371(CHEMBL4457285)
Affinity DataIC50: 6.05E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515360(CHEMBL4459519)
Affinity DataIC50: 7.13E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515356(CHEMBL4442901)
Affinity DataIC50: 7.31E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515358(CHEMBL4553319)
Affinity DataIC50: 9.61E+3nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515361(CHEMBL4513369)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515359(CHEMBL4563821)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515364(CHEMBL4557687)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515357(CHEMBL4586100)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515355(CHEMBL4591546)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515352(CHEMBL4568512)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515346(CHEMBL4470913)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515370(CHEMBL4522651)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p300 (unknown origin) using biotinylated histone H3 (1 to 21 residues) as substrate measured after 90 mins in presence of Acetyl CoA by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515347(CHEMBL4461759)
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of recombinant HDAC6 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515347(CHEMBL4461759)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant HDAC8 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515347(CHEMBL4461759)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant HDAC2 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515347(CHEMBL4461759)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50515347(CHEMBL4461759)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant HDAC3 (unknown origin) measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed