Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50008212
TargetProstaglandin G/H synthase 2(Human)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50516770(CHEMBL4444717)
Affinity DataIC50: 22nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50516768(CHEMBL4456822)
Affinity DataIC50: 23nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50516769(CHEMBL4438795)
Affinity DataIC50: 23nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50516767(CHEMBL4591824)
Affinity DataIC50: 32nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50516769(CHEMBL4438795)
Affinity DataIC50: 195nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50516770(CHEMBL4444717)
Affinity DataIC50: 312nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50516767(CHEMBL4591824)
Affinity DataIC50: 361nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50516768(CHEMBL4456822)
Affinity DataIC50: 407nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 490nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 500nMAssay Description:Inhibition of ovine COX-1 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Anhui University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of human COX-2 using arachidonic acid as substrate incubated for 5 mins by fluorescence-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)