Compile Data Set for Download or QSAR
Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 50008407
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518977(CHEMBL1160734)
Affinity DataKd:  0.891nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataKd:  1.40nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataKd:  1.5nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM25759([3-(9H-carbazol-4-yloxy)-2-hydroxypropyl][2-(2-met...)
Affinity DataKd:  0.195nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518981(CHEMBL4594173)
Affinity DataKd:  1.30nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518978(CHEMBL4446394)
Affinity DataKd:  1.90nMAssay Description:Displacement of [3H]DHA from beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518977(CHEMBL1160734)
Affinity DataIC50: 0.724nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518969(CHEMBL4514723)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518981(CHEMBL4594173)
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518984(CHEMBL4564189)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518978(CHEMBL4446394)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518985(CHEMBL4465278)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518984(CHEMBL4564189)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518982(CHEMBL4462252)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518974(CHEMBL4574652)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518972(CHEMBL1395661)
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518977(CHEMBL1160734)
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518993(CHEMBL4527821)
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518969(CHEMBL4514723)
Affinity DataIC50: 2.90nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518973(CHEMBL4473518)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518975(CHEMBL4450606)
Affinity DataIC50: 3.30nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518979(CHEMBL4434772)
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518973(CHEMBL4473518)
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518990(CHEMBL4532142)
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518982(CHEMBL4462252)
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518969(CHEMBL4514723)
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518993(CHEMBL4527821)
Affinity DataIC50: 5.20nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataIC50: 5.5nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518985(CHEMBL4465278)
Affinity DataIC50: 5.60nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518966(CHEMBL4515576)
Affinity DataIC50: 5.90nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518977(CHEMBL1160734)
Affinity DataIC50: 5.90nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518976(CHEMBL4442559)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518986(CHEMBL4584173)
Affinity DataIC50: 6.5nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518981(CHEMBL4594173)
Affinity DataIC50: 6.60nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518968(CHEMBL4441975)
Affinity DataIC50: 6.90nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518978(CHEMBL4446394)
Affinity DataIC50: 7.60nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518980(CHEMBL4459989)
Affinity DataIC50: 8.30nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518979(CHEMBL4434772)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518987(CHEMBL4472564)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518967(CHEMBL4530266)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518968(CHEMBL4441975)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518988(CHEMBL4593049)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518984(CHEMBL4564189)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518991(CHEMBL4564495)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518979(CHEMBL4434772)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) expressed in HEK293 cell assessed as inhibition of isoproterenol-induced cAMP produ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518974(CHEMBL4574652)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518982(CHEMBL4462252)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518993(CHEMBL4527821)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
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