Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50008208
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
S£O Paulo State University

Curated by ChEMBL
LigandPNGBDBM255614(US9499570, D140)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of full-length human recombinant PDE4B catalytic domain (152 to 484 residues)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
S£O Paulo State University

Curated by ChEMBL
LigandPNGBDBM50516760(CHEMBL4526356)
Affinity DataIC50: 4.10nMAssay Description:Selective estrogen receptor down regulator activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
S£O Paulo State University

Curated by ChEMBL
LigandPNGBDBM50516758(CHEMBL4444471 | US11542283, Compound V-9A)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human chymotrypsin-like activity of 20S proteasome (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
S£O Paulo State University

Curated by ChEMBL
LigandPNGBDBM50516762(CHEMBL4474485)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human neutrophil ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
S£O Paulo State University

Curated by ChEMBL
LigandPNGBDBM50516759(CHEMBL4458610)
Affinity DataKi:  17nMAssay Description:Inhibition of human chymotrypsin-like activity of 20S proteasome (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetBeta-lactamase TEM(Escherichia coli)
S£O Paulo State University

Curated by ChEMBL
LigandPNGBDBM50516761(CHEMBL3286879)
Affinity DataKi:  40nMAssay Description:Inhibition of bacterial beta lactamase TEM-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed