Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50006684
TargetToll-like receptor 8(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50502464(CHEMBL1443979)
Affinity DataIC50: 9.20E+3nMAssay Description:Antagonist activity at human TLR8 expressed in HEK-Blue cells assessed as inhibition of CL075-induced NF-kappaB activation incubated for 1 hr followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetToll-like receptor 8(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50502465(CHEMBL1401818)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human TLR8 expressed in HEK-Blue cells assessed as inhibition of CL075-induced NF-kappaB activation incubated for 1 hr followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetToll-like receptor 8(Human)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50502466(CHEMBL4589214)
Affinity DataIC50: 3.55E+4nMAssay Description:Antagonist activity at human TLR8 expressed in HEK-Blue cells assessed as inhibition of CL075-induced NF-kappaB activation incubated for 1 hr followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed