Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50008055
TargetToll-like receptor 4(Human)
Ajou University

Curated by ChEMBL
LigandPNGBDBM50515277(CHEMBL4436411)
Affinity DataKd:  1.40nMAssay Description:Binding affinity to recombinant human TLR4 assessed as dissociation constant up to 200 uM by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLymphocyte antigen 96(Human)
Ajou University

Curated by ChEMBL
LigandPNGBDBM50515277(CHEMBL4436411)
Affinity DataKd:  2.40nMAssay Description:Binding affinity to recombinant human MD2 assessed as dissociation constant up to 200 uM by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetToll-like receptor 4(Human)
Ajou University

Curated by ChEMBL
LigandPNGBDBM50515276(CHEMBL4463337)
Affinity DataKd:  1.10nMAssay Description:Binding affinity to recombinant human TLR4 assessed as dissociation constant up to 200 uM by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLymphocyte antigen 96(Human)
Ajou University

Curated by ChEMBL
LigandPNGBDBM50515276(CHEMBL4463337)
Affinity DataKd:  4.90nMAssay Description:Binding affinity to recombinant human MD2 assessed as dissociation constant up to 200 uM by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetToll-like receptor 4(Human)
Ajou University

Curated by ChEMBL
LigandPNGBDBM50515277(CHEMBL4436411)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at TLR4 (unknown origin) assessed as inhibition of proinflammatory cytokinesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetToll-like receptor 4(Human)
Ajou University

Curated by ChEMBL
LigandPNGBDBM50515276(CHEMBL4463337)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at TLR4 (unknown origin) assessed as inhibition of proinflammatory cytokinesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetToll-like receptor 4(Human)
Ajou University

Curated by ChEMBL
LigandPNGBDBM50515277(CHEMBL4436411)
Affinity DataIC50: 2.50E+4nMAssay Description:Antagonist activity at TLR4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetToll-like receptor 4(Human)
Ajou University

Curated by ChEMBL
LigandPNGBDBM50515276(CHEMBL4463337)
Affinity DataIC50: 4.00E+4nMAssay Description:Antagonist activity at TLR4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed