Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50010154
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50535681(CHEMBL4438095)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human Kv7.2/Kv7.3 expressed in CHO cells at holding potential of at -85 mV by whole cell patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50535682(CHEMBL4580661)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human Kv7.2/Kv7.3 expressed in CHO cells at holding potential of at -85 mV by whole cell patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed