Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50007769
TargetP2Y purinoceptor 14(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50343877(7-(4-fluoro-2,6-dimethylbenzyloxy)-4-(thiophen-3-y...)
Affinity DataIC50: 14nMAssay Description:Inhibition of mouse P2Y14 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50512416(CHEMBL4447162)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of human P2Y14 receptor expressed in CHO cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50343888((R)-4-(4-(2,2-difluoro-1-hydroxyethyl)phenyl)-7-(4...)
Affinity DataKi:  4nMAssay Description:Inhibition of mouse P2Y14 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataKi:  35nMAssay Description:Inhibition of mouse P2Y14 receptor in presence of 2% HSAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50343888((R)-4-(4-(2,2-difluoro-1-hydroxyethyl)phenyl)-7-(4...)
Affinity DataKi:  1.29E+3nMAssay Description:Inhibition of mouse P2Y14 receptor in presence of 2% HSAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed