Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50007752
TargetProstaglandin G/H synthase 2(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM222462((E)-4-[4-(2-Chlorobenzylidene)-2-(4-chlorophenyl)-...)
Affinity DataIC50: 860nMAssay Description:Inhibition of recombinant human COX2 by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetProbable maltase-glucoamylase 2(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50502118(CHEMBL4476702)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl-a-d-glucopyranoside as substrate preincubated for 5 mins followed by substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM222462((E)-4-[4-(2-Chlorobenzylidene)-2-(4-chlorophenyl)-...)
Affinity DataIC50: 7.86E+3nMAssay Description:Inhibition of ovine COX1 by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50512315(CHEMBL4438040)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBeta-glucuronidase(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM178133(3-(6-Chloro-1H-imidazo[4,5-b]pyridin-2-yl)benzene-...)
Affinity DataIC50: 2.93E+4nMAssay Description:Inhibition of beta-glucuronidase (unknown origin) using p-nitrophenyl-beta-D-glucuronide as substrate pre-incubated for 30 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed