Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50008963
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM430732(US10544150, Compound 115 | (R)-(4-fluorophenyl)(8-...)
Affinity DataIC50: 260nMAssay Description:Antagonistic activity against NK3R (unknown origin) expressed in CHO cells assessed as inhibition of NKB-induced intracellular calcium flux by Calciu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50524029(CHEMBL4567857)
Affinity DataIC50: 4.10E+3nMAssay Description:Antagonistic activity against NK3R (unknown origin) expressed in CHO cells assessed as inhibition of NKB-induced intracellular calcium flux by Calciu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50524033(CHEMBL4558106)
Affinity DataIC50: 8.20E+3nMAssay Description:Antagonistic activity against NK3R (unknown origin) expressed in CHO cells assessed as inhibition of NKB-induced intracellular calcium flux by Calciu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50524032(CHEMBL4569878)
Affinity DataIC50: 1.03E+4nMAssay Description:Antagonistic activity against NK3R (unknown origin) expressed in CHO cells assessed as inhibition of NKB-induced intracellular calcium flux by Calciu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50524031(CHEMBL4437427)
Affinity DataIC50: 1.18E+4nMAssay Description:Antagonistic activity against NK3R (unknown origin) expressed in CHO cells assessed as inhibition of NKB-induced intracellular calcium flux by Calciu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50524030(CHEMBL4516772)
Affinity DataIC50: 1.37E+4nMAssay Description:Antagonistic activity against NK3R (unknown origin) expressed in CHO cells assessed as inhibition of NKB-induced intracellular calcium flux by Calciu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50524032(CHEMBL4569878)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonistic activity against NK3R (unknown origin) expressed in CHO cells assessed as inhibition of NKB-induced intracellular calcium flux under UV-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed