Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50007490
TargetDual specificity protein kinase CLK1(Mouse)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50509920(CHEMBL4558273)
Affinity DataIC50: 87nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacteria using GRSRSRSRSRSR as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50509919(CHEMBL4465324)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CLK1 (129 to end residues) expressed in baculovirus infected Sf9 insect cells sing MBP as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50509919(CHEMBL4465324)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of recombinant full-length rat N-terminal GST-tagged DYRK1A was expressed in Escherichia coli using DYRKtide as substrate measured after 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed