Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50010329
TargetSolute carrier family 22 member 8(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537500(CHEMBL4562825)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 8(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537497(CHEMBL4519013)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 8(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537498(CHEMBL4584575)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 8(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537496(CHEMBL4527448)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 8(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537501(CHEMBL4582456)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537496(CHEMBL4527448)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537500(CHEMBL4562825)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 8(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537502(CHEMBL38650 | NSC-220968)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 8(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537499(CHEMBL4525573)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537498(CHEMBL4584575)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537497(CHEMBL4519013)
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 8(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50180512(1-methyl-5-vinyl-9,10-dihydrophenanthrene-2,7-diol...)
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of OAT3 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50180512(1-methyl-5-vinyl-9,10-dihydrophenanthrene-2,7-diol...)
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50537499(CHEMBL4525573)
Affinity DataIC50: 4.31E+4nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed