Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50007899
TargetKallikrein-7(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513785(CHEMBL4575658)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human KLK7 expressed in expressed in Pichia pastoris X-33 cells using KHLY-pNA as susbtrate measured every 15 secs for 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513785(CHEMBL4575658)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human matriptase using Boc-QAR-MCA as susbtrate measured every 60 secs for 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513781(CHEMBL4466351)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human matriptase using Boc-QAR-MCA as susbtrate measured every 60 secs for 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-7(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513781(CHEMBL4466351)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human KLK7 expressed in expressed in Pichia pastoris X-33 cells using KHLY-pNA as susbtrate measured every 15 secs for 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-7(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513783(CHEMBL4456620)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human KLK7 expressed in expressed in Pichia pastoris X-33 cells using KHLY-pNA as susbtrate measured every 15 secs for 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-7(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513780(CHEMBL4456106)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant KLK7 (unknown origin) expressed in Pichia pastoris X-33 cells using p-NA peptide as substrate measured every 10 secs for 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513783(CHEMBL4456620)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human matriptase using Boc-QAR-MCA as susbtrate measured every 60 secs for 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513781(CHEMBL4466351)
Affinity DataKi:  0.340nMAssay Description:Inhibition of recombinant human KLK5 expressed in expressed in Pichia pastoris X-33 cells using Boc-VPR-MCA as susbtrate measured every 60 secs for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513784(CHEMBL4550494)
Affinity DataKi:  0.730nMAssay Description:Inhibition of recombinant human KLK5 expressed in expressed in Pichia pastoris X-33 cells using Boc-VPR-MCA as susbtrate measured every 60 secs for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513785(CHEMBL4575658)
Affinity DataKi:  2.40nMAssay Description:Inhibition of recombinant human KLK5 expressed in expressed in Pichia pastoris X-33 cells using Boc-VPR-MCA as susbtrate measured every 60 secs for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513783(CHEMBL4456620)
Affinity DataKi:  3.70nMAssay Description:Inhibition of recombinant human KLK5 expressed in expressed in Pichia pastoris X-33 cells using Boc-VPR-MCA as susbtrate measured every 60 secs for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513782(CHEMBL4513520)
Affinity DataKi:  8.90nMAssay Description:Inhibition of recombinant human KLK5 expressed in expressed in Pichia pastoris X-33 cells using Boc-VPR-MCA as susbtrate measured every 60 secs for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-14(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513781(CHEMBL4466351)
Affinity DataKi:  18nMAssay Description:Inhibition of recombinant human KLK14 expressed in Spodoptera frugiperda Sf9 cells using Boc-QAR-MCA as susbtrate measured every 60 secs for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-14(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513780(CHEMBL4456106)
Affinity DataKi:  25nMAssay Description:Inhibition of recombinant KLK14 (unknown origin) expressed in Spodoptera frugiperda Sf9 cells using pNA peptide as susbtrate measured every 10 secs f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-14(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513783(CHEMBL4456620)
Affinity DataKi:  79nMAssay Description:Inhibition of recombinant human KLK14 expressed in Spodoptera frugiperda Sf9 cells using Boc-QAR-MCA as susbtrate measured every 60 secs for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513780(CHEMBL4456106)
Affinity DataKi:  143nMAssay Description:Inhibition of recombinant KLK5 (unknown origin) expressed in Pichia pastoris X-33 cells using pNA peptide as susbtrate measured every 10 secs for 300...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetKallikrein-14(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513785(CHEMBL4575658)
Affinity DataKi:  150nMAssay Description:Inhibition of recombinant human KLK14 expressed in Spodoptera frugiperda Sf9 cells using Boc-QAR-MCA as susbtrate measured every 60 secs for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSuppressor of tumorigenicity 14 protein(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50513780(CHEMBL4456106)
Affinity DataKi:  200nMAssay Description:Inhibition of recombinant human matriptase catalytic domain using Boc-QARAMC as substrate preincubated for 1 hr followed by substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed